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Streamlined strategy for discovering active compounds for nephrolithiasis treatment from herbal medicines using the fruit fly model

Bibliographic Data

ID14744719
AuthorsYunuo Ren (Tianjin University, corresponding author), Wen Zhang (0000-0002-8166-2879), Wen Jie Zhang (0009-0007-6671-0637, Tianjin University), Youxin Li (0000-0002-0812-744X, Tianjin University), Dekun Wang (0000-0002-1779-8376, Nankai University), Weiwei Tang (0000-0002-0725-3073, Tianjin University), Lingfei Wang (0000-0001-7046-9478, First Teaching Hospital of Tianjin University of Traditional Chinese Medicine), Xinghua Jin (0000-0002-8883-5234, Tianjin University), Donghai Xia (Dalian Institute of Chemical Physics), Wei Yu (0000-0003-1933-5380), Yu Wei (0000-0003-3809-1449, Dalian Institute of Chemical Physics), Yaodong Miao (0000-0002-6627-5694, Tianjin University of Traditional Chinese Medicine), Yingjie Ju (0000-0001-8833-8441, Tianjin University), Shushen Sun, Shixiang Sun (0000-0001-5499-2963, Tianjin Hospital), Tianxiang Li (0009-0004-3460-8361, Tianjin University of Traditional Chinese Medicine), Shaoshan Du, Shiyu Du (0000-0001-6707-3915, Tianjin Hospital), Zhimou Guo (0000-0001-7129-186X, Dalian Institute of Chemical Physics), Xiaoyue Tan (0000-0001-9989-0573, Nankai University), Zhiguang Yuchi (0000-0003-2595-9106, Tianjin University of Science and Technology), Yiwen Wang (0000-0002-6879-8974, Tianjin University)
Year2025
Volume348
Pages119846
Publication date2025-05-01
Open AccessYes
TypeARTICLE
VenueJournal of Ethnopharmacology (JOURNAL)
Journal identifiersISSN: 0378-8741 • E-ISSN: 1872-7573
PublisherElsevier BV (PUBLISHER)
DOI10.1016/j.jep.2025.119846
PMID40280373
OpenAlexW4409728769
LanguageEN
References cited33

We developed an efficient strategy for identifying core components of TCMs for kidney stones treatment using a fruit fly model combined with chemical isolation and identification techniques. This approach led to the discovery of three novel potential compounds for controlling kidney stones. Validated in mammalian models, these findings underscore the fruit fly model's utility in uncovering bioactive substances from TCMs, laying the groundwork for future research and the development of novel kidney stones therapies

Alternative medicine · Biological activity · Biology · Pharmacognosy · Phytotherapy · Traditional medicine · Cassava research and cyanide · Heavy Metals in Plants · Kidney Stones and Urolithiasis Treatments · Medicine · Biochemistry · Pharmacology

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